Publications
Recent publications from the group
Synthesis and Biological Evaluation of Colchicine – Aryl/ alkyl amine Hybrids as Potential Non-cytotoxic Cholinesterase Inhibitors: Identification of SBN-284 as a Dual Inhibitor of Cholinesterases and NLRP3 Inflammasome
Reddy CN, Nuthakki VK, Sharma A, Malik S, Tabassum B, Kumar R, Choudhary S, Iqbal F, Tufail Z, Mondhe DM, Kumar A, Bharate SB*
ACS Chem. Neurosci., 2024, 15, 2779–2794
Structure-Based Virtual Screening of FDA-approved Drugs to Discover Potential Inhibitors of Phosphoinositide Kinase, PIKfyve
Wadje BN, Somarowthu T, Thakur S, Jadhav HR, Bharate SB*
J. Biomol. Struct. Dyn. 2024, In Press
EDITORIAL: Natural Products Driven Medicinal Chemistry
Bharate SB and Lindsley CW
J. Med. Chem. 2023, 66, 24, 16455–16456
Design, Synthesis, and Pharmacological Evaluation of Embelin-Aryl/alkyl amine Hybrids as Orally Bioavailable Blood-Brain Barrier Permeable Multitargeted Agents with Therapeutic Potential in Alzheimer's Disease: Discovery of SB-1448
Nuthakki VK, Choudhary S, Reddy CN, Bhatt S, Jamwal A, Jotshi A, Raghuvanshi, R, Sharma A, Thakur S, Jadhav H, Bharate SS, Nandi U, Kumar A, Bharate SB*
ACS Chem Neurosci. 2023, 14, 6, 1193–1219
Cell-intrinsic Aryl Hydrocarbon Receptor signalling is required for the resolution of injury-induced colonic stem cells
Shah K, Maradana MR, Delás MJ, Metidji A, Graelmann F, Llorian M, Chakravarty P, Li Y, Tolaini M, Shapiro M, Kelly G, Cheshire C, Bhurta D, Bharate SB, Stockinger B.
Nature Commun. 2022, 13 (1), 1827
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